Free shipping on all orders over $ 500

GR 113808

Cat. No. M6759

All AbMole products are for research use only, cannot be used for human consumption.

GR 113808 Structure
Size Price Availability
5mg USD 90  USD90 Out of stock
10mg USD 150  USD150 Out of stock
Free Delivery on orders over USD 500 Bulk Inquiry?

Quality Control & Documentation
Biological Activity

GR 113808 is a potent, selective 5-HT4 receptor antagonist (pKB = 9.43 in human colonic muscle, and Kd = 0.15 nM for binding to cloned human 5-HT4 receptors). Displays > 300-fold selectivity over 5-HT1A, 5-HT1B, 5-HT2A, 5-HT2C and 5-HT3 receptors.

Chemical Information
Molecular Weight 393.5
Formula C19H27N3O4S
CAS Number 144625-51-4
Form Solid
Solubility (25°C) 1eq. HCl 9.84 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Outeiro, et al. Science. Sirtuin 2 inhibitors rescue α-synuclein-mediated toxicity in models of Parkinson's disease.

Related 5-HT Receptor Products
Aripiprazole-d8

Aripiprazole-d8

Clozapine-d8

Clozapine-d8

Olanzapine-d3

Olanzapine-d3

Quetiapine-d8 fumarate

Quetiapine-d8 fumarate

Dapoxetine hydrochloride-d7

Dapoxetine hydrochloride-d7

  Catalog
Abmole Inhibitor Catalog




Keywords: GR 113808 supplier, 5-HT Receptor, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.



Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.