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GlyH 101

Cat. No. M6754

All AbMole products are for research use only, cannot be used for human consumption.

GlyH 101 Structure
Synonym:

GlyH101

Size Price Availability Quantity
Free Sample (0.5-1 mg)  USD 0 In stock
2mg USD 60  USD60 In stock
5mg USD 90  USD90 In stock
10mg USD 170  USD170 In stock
25mg USD 340  USD340 In stock
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Quality Control & Documentation
Biological Activity

GlyH 101 is a reversible, voltage-dependent CFTR chloride channel blocker (Ki = 4.3 μM). Inhibits forskolin-induced hyperpolarization in nasal potential differences and inhibits cholera toxin-induced intestinal fluid secretion in mice.

Chemical Information
Molecular Weight 493.15
Formula C19H15Br2N3O3
CAS Number 328541-79-3
Solubility (25°C) DMSO 49.31 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Smedt, et al. CNS Drug Rev. Levetiracetam: the profile of a novel anticonvulsant drug - part I: preclinical data.

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Keywords: GlyH 101, GlyH101 supplier, CFTR, inhibitors, activators

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