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Gepirone

Cat. No. M40960

All AbMole products are for research use only, cannot be used for human consumption.

Gepirone Structure
Synonym:

BMY-13805

Size Price Availability Quantity
5mg USD 59  USD59 In stock
10mg USD 89  USD89 In stock
25mg USD 149  USD149 In stock
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Quality Control & Documentation
Biological Activity

Gepirone (Gepirone) is a first-in-class, selective, affinity-based, orally active 5-HT1A receptor partial agonist as well as a 5-HT2A receptor antagonist for use in studies related to anxiety, depression, and chronic kidney disease.

Chemical Information
Molecular Weight 359.47
Formula C19H29N5O2
CAS Number 83928-76-1
Form Solid
Storage 4°C, protect from light
References

[1] A Kaur Gill et al. Drugs Today (Barc). Gepirone hydrochloride: a novel antidepressant with 5-HT1A agonistic properties

[2] Donald S Robinson et al. Clin Ther. A review of the efficacy and tolerability of immediate-release and extended-release formulations of gepirone

[3] R A Leslie. Curr Opin Investig Drugs. Gepirone. Organon

[4] J P Yevich et al. Prog Clin Biol Res. Gepirone hydrochloride: preclinical pharmacology and recent clinical findings

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Keywords: Gepirone, BMY-13805 supplier, 5-HT Receptor, inhibitors, activators

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