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Frovatriptan Succinate

Cat. No. M20943

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Frovatriptan Succinate Structure

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Quality Control & Documentation
Biological Activity

Frovatriptan Succinate is the succinate salt form of frovatriptan, a synthetic triptan with serotonin (5-HT) receptor agonist activity especially for the 5-HT1B/1D receptors.

Chemical Information
Molecular Weight 361.39
Formula C18H23N3O5
CAS Number 158930-09-7
Solubility (25°C) DMSO 72 mg/mL
Water 72 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Hongquan Zheng, et al. Drug Des Devel Ther. Pharmacokinetic Study of Frovatriptan Succinate Tablet After Single and Multiple Oral Doses in Chinese Healthy Subjects

[2] Roemer B Brandt, et al. CNS Drugs. Pharmacotherapy for Cluster Headache

[3] No authors listed. Frovatriptan

[4] S D Silberstein, et al. Neurology. Evidence-based guideline update: pharmacologic treatment for episodic migraine prevention in adults: report of the Quality Standards Subcommittee of the American Academy of Neurology and the American Headache Society

[5] E A Balbisi. Int J Clin Pract. Frovatriptan succinate, a 5-HT1B/1D receptor agonist for migraine

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Keywords: Frovatriptan Succinate supplier, 5-HT Receptor, inhibitors, activators

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