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Etavopivat

Cat. No. M21076

All AbMole products are for research use only, cannot be used for human consumption.

Etavopivat Structure
Synonym:

FT-4202

Size Price Availability Quantity
1mg USD 200  USD200 In stock
5mg USD 480  USD480 In stock
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Biological Activity

Etavopivat, an oral erythrocyte pyruvate kinase (PKR) activator, is being developed for sickle cell disease and other hemoglobinopathies, previously reported in 2019.

Chemical Information
Molecular Weight 457.50
Formula C22H23N3O6S
CAS Number 2245053-57-8
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Bruno Fattizzo, et al. Front Med (Lausanne). Rise of the planet of rare anemias: An update on emerging treatment strategies

[2] Patricia Schroeder, et al. J Pharmacol Exp Ther. Etavopivat, a Pyruvate Kinase Activator in Red Blood Cells, for the Treatment of Sickle Cell Disease

[3] Sanjeev Forsyth, et al. Clin Pharmacol Drug Dev. Safety, Pharmacokinetics, and Pharmacodynamics of Etavopivat (FT-4202), an Allosteric Activator of Pyruvate Kinase-R, in Healthy Adults: A Randomized, Placebo-Controlled, Double-Blind, First-in-Human Phase 1 Trial

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  Catalog
Abmole Inhibitor Catalog




Keywords: Etavopivat, FT-4202 supplier, Pyruvate Kinase, inhibitors, activators

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