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EN40 

Cat. No. M29205

All AbMole products are for research use only, cannot be used for human consumption.

EN40  Structure

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Quality Control & Documentation
Biological Activity

EN40 is a potent, selective aldehyde dehydrogenase 3A1 (ALDH3A1) inhibitor as a covalent ligand, exhibits an IC50 value of 2 uM.

*The compound is unstable in solutions, freshly prepared is recommended

Chemical Information
Molecular Weight 217.26
Formula C13H15NO2
CAS Number 2094547-67-6
Form Oil
Solubility (25°C) DMSO 5 mg/mL (ultrasonic)
Ethanol 2 mg/mL (ultrasonic)
Storage 4°C, sealed
References

[1] Jessica L Counihan, et al. ACS Chem Biol. Chemoproteomics-Enabled Covalent Ligand Screening Reveals ALDH3A1 as a Lung Cancer Therapy Target

[2] S Tang, et al. Anim Genet. A novel 62-bp indel mutation in the promoter region of transforming growth factor-beta 2 (TGFB2) gene is associated with body weight in chickens

[3] P Beau, et al. Clin Nutr. Cholesterol-lowering effect of continuous enteral nutrition in man

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  Catalog
Abmole Inhibitor Catalog




Keywords: EN40  supplier, ALDH, inhibitors, activators

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