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DPH binds and alters the conformation of the myristoyl binding site of c-Abl tyrosine kinase. It exhibits potent enzymatic and cellular activity that stimulates the activation of c-Abl.
| Molecular Weight | 336.32 |
| Formula | C18H13FN4O2 |
| CAS Number | 484049-04-9 |
| Solubility (25°C) | DMSO 45 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[4] Jarmila Repkov, et al. Influence of DPH on the structure and dynamics of a DPPC bilayer
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