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Cyclobuxine D

Cat. No. M18968

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Cyclobuxine D Structure

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Quality Control & Documentation
Biological Activity

Cyclobuxine D has a significant bradycardic effect in the rat heart and an inhibitory action on acetylcholine and Ba++−induced contraction of the longitudinal muscle isolated from the rabbit jejunum.

Chemical Information
Molecular Weight 386.61
Formula C25H42N2O
CAS Number 2241-90-9
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] H R MAHLER, et al. J Mol Biol. NUCLEIC ACID INTERACTIONS. V. EFFECTS OF CYCLOBUXINE

[2] J H Lee, et al. Planta Med. Cyclobuxine protects the isolated rat heart from the myocardial injuries produced by ischemia and reperfusion

[3] D Herlem-Gaulier, et al. Bull Soc Chim Fr. [Steroid alkaloids. LVI. Family of Buxaceae. (8.) Alkaloids of Buxus balearica: structure of N-3-isobutyryl cyclobuxine-F (baleabuxine)]

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Keywords: Cyclobuxine D supplier, AChR/AChE, inhibitors, activators

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