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CRT0273750

Cat. No. M10809

All AbMole products are for research use only, cannot be used for human consumption.

CRT0273750 Structure

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Quality Control & Documentation
Biological Activity

CRT0273750 is a lead compound of autotaxin (ATX) inhibitors and regulates plasma LPA levels. CRT0273750 can be used in ATX/LPA dependent cancer models.

Chemical Information
Molecular Weight 502.92
Formula C25H22ClF3N4O2
CAS Number 1979939-16-6
Solubility (25°C) DMSO ≥ 200 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Pritom Shah, et al. Bioorg Med Chem Lett. Discovery of potent inhibitors of the lysophospholipase autotaxin

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  Catalog
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Keywords: CRT0273750 supplier, PDE, inhibitors, activators

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