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CP-628006

Cat. No. M21215

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CP-628006  Structure
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Biological Activity

CP-628006 is a CFTR small molecule enhancer that enhances CFTR function in human bronchial epithelial (hBE) cells and restores ATP-dependent gated channels in cystic fibrosis mutant G551D-CFTR. It can be used in cystic fibrosis (CF) related studies.

Chemical Information
Molecular Weight 536.63
Formula C32H35F3N2O2
CAS Number 305822-08-6
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Jia Liu, et al. Br J Pharmacol. A small molecule CFTR potentiator restores ATP-dependent channel gating to the cystic fibrosis mutant G551D-CFTR

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Keywords: CP-628006 supplier, CFTR, inhibitors, activators

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