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Cerlapirdine (SAM-531, PF-05212365) is a selective and potent full antagonist of the 5-hydroxytryptamine 6 (5-HT6) receptor. Cerlapirdine has the potential for researching the Alzheimer's disease.
| Molecular Weight | 409.5 |
| Formula | C22H23N3O3S |
| CAS Number | 925448-93-7 |
| Form | Solid |
| Solubility (25°C) | DMSO 41.67 mg/mL (ultrasonic and warming and adjust pH to 3 with HCl and heat to 60°C) |
| Storage | 4°C, protect from light |
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