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BRCA1-IN-2

Cat. No. M9864

All AbMole products are for research use only, cannot be used for human consumption.

BRCA1-IN-2 Structure
Synonym:

BRCA1-IN II

Size Price Availability
5mg USD 480  USD480 4-7 Days
10mg USD 800  USD800 4-7 Days
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Quality Control & Documentation
Biological Activity

BRCA1-IN-2 is a cell-permeable protein-protein interaction (PPI) inhibitor for BRCA1, with IC50 of 0.31 μM and Kd of 0.3 μM. BRCA1-IN-2 has antitumor activities via the disruption of BRCA1 (BRCT)2/protein interactions.

Chemical Information
Molecular Weight 544.54
Formula C26H33N4O7P
CAS Number 1622262-55-8
Solubility (25°C) DMSO
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Zhenkun Na, et al. Methods Mol Biol. Protein-Protein Interaction Inhibitors of BRCA1 Discovered Using Small Molecule Microarrays

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  Catalog
Abmole Inhibitor Catalog




Keywords: BRCA1-IN-2, BRCA1-IN II supplier, PARP, inhibitors, activators

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