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AU-15330 is a protein hydrolysis-targeted chimeric (PROTAC) degradation of SWI/SNF ATPase subunits SMARCA2 and SMARCA4, and also induces effective tumor growth inhibition in a prostate cancer xenograft model.
| Molecular Weight | 755.94 |
| Formula | C39H49N9O5S |
| CAS Number | 2380274-50-8 |
| Form | Solid |
| Solubility (25°C) | DMSO >140 mg/mL |
| Storage | 4°C, dry |
[2] Lanbo Xiao, et al. Nature. Targeting SWI/SNF ATPases in enhancer-addicted prostate cancer
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