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ALK4290

Cat. No. M28040

All AbMole products are for research use only, cannot be used for human consumption.

ALK4290 Structure
Synonym:

AKST4290

Price and Availability

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Quality Control & Documentation
Biological Activity

ALK4290 (AKST4290) is a potent and orally active CCR3 inhibitor, with a Ki of 3.2 nM for hCCR3. ALK4290 can be used for the research of neovascular age-related macular degeneration and Parkinsonism.

Chemical Information
Molecular Weight 512.04
Formula C27H34ClN5O3
CAS Number 1251528-23-0
Form Solid
Solubility (25°C) DMSO 50 mg/mL (ultrasonic and warming and heat to 60°C)
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Michael W Stewart, et al. Retina. SAFETY AND THERAPEUTIC EFFECTS OF ORALLY ADMINISTERED AKST4290 IN NEWLY DIAGNOSED NEOVASCULAR AGE-RELATED MACULAR DEGENERATION

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  Catalog
Abmole Inhibitor Catalog




Keywords: ALK4290, AKST4290 supplier, CCR, inhibitors, activators

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