| Cat.No. | Name | Information |
|---|---|---|
| M9573 | Orexin A (human, mouse, rat, bovine) | Orexin A (human, mouse, rat, bovine) is a specific, high-affinity agonist for G-protein-coupled receptor OX1R. |
| M3261 | Almorexant | Almorexant is a competitive OX1 and OX2 orexin receptor antagonist with IC50 of 13 and 8 nM, respectively. |
| M6833 | IPSU | IPSU is a oX 2 receptor antagonist; orally bioavailable. |
| M3796 | SB-334867 hydrochloride | SB-334867 hydrochloride is a selective non-peptide orexin OX1 receptor antagonist with a pKb value of 7.2. |
| M3760 | TCS-1102 | TCS 1102 is a potent, dual orexin receptor antagonist (Ki values are 0.2 and 3 nM for OX2 and OX1 receptors respectively). |
| M3710 | MK-3697 | MK-3697 is an isonicotinamide small molecule, acting as a potent and selective Orexin 2 receptor antagonist with Ki = 0.95 nM. |
| M3324 | SB408124 | SB408124 (Tocris-1963) is a non-peptide antagonist for OX1 receptor with Ki of 57 nM and27 nM in both whole cell and membrane, respectively, exhibits 50-fold selectivity over OX2 receptor. |
| M2124 | MK-6096 | MK-6096 is an orally bioavailable potent and selective reversible antagonist of OX(1)R and OX(2)R. |
| M56300 | CVN766 | CVN766 is an orally active inhibitor of orexin 1 receptor antagonist with blood-brain permeability with the IC50 values of 8 nM and >10 μM for OX1R and OX2R, respectively. |
| M56299 | Nivasorexant | Nivasorexant is a potent orexin receptor antagonist. |
| M54494 | [Ala11, D-Leu15]-Orexin B(human) | [Ala11,D-Leu15]-Orexin B(human) is a potent and selective orexin-2 receptor (OX2) agonist. |
| M54469 | Orexin B, rat, mouse | Orexin B, rat, mouse (Rat orexin B) is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively. |
| M52942 | Hypocretin (70-98), human | Hypocretin (70-98), human is a polypeptide that is capable of binding to an orexin receptor OX1R and promotes apoptosis. |
| M52941 | Xenopus orexin A | Xenopus orexin A is a neuropeptides that identified as an endogenous ligands for an orphan G-protein-coupled receptor. |
| M52940 | Xenopus orexin B | Xenopus orexin B is a neuropeptides that identified as an endogenous ligands for an orphan G-protein-coupled receptor. |
| M52939 | Orexin B, human | Orexin B, human is an endogenous agonist at Orexin receptor with Kis of 420 and 36 nM for OX1 and OX2, respectively. |
| M50234 | CVN766 | CVN766 is an oral small molecule orexin 1 receptor (Ox1R) antagonist that is approximately 1000 times more selective for Ox1R than Ox2R. |
| M41898 | Orexin receptor modulator-1 | Orexin receptor modulator-1 is an orexin receptor modulator. |
| M41897 | RTIOXA-43 | RTIOXA-43 is a orexin receptor agonist with EC50s of 24 nM and 24 nM for OX2 and OX1 receptors, respectively. |
| M41896 | Firazorexton hydrate | Firazorexton hydrate (TAK-994) is a potent, brain-penetrant, and orally active orexin type 2 receptor (OX2R) agonist (EC50: 19 nM). |
| M29477 | Firazorexton | Firazorexton is a potent orexin type 2 receptor (OX2R) agonist. |
| M29476 | Suntinorexton | Suntinorexton, a heterocyclic compound, is an orexin type 2 receptor agonist. |
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