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IPSU is a oX2 receptor antagonist. Exhibits approximately six-fold selectivity for OX2 versus OX1 receptors. Decreases activity and increases sleep time in mice during the active phase, without affecting REM/NREM balance. Orally bioavailable. Brain penetrant.
| Molecular Weight | 405.49 |
| Formula | C23H27N5O2 |
| CAS Number | 1373765-19-5 |
| Form | Solid |
| Solubility (25°C) | 1eq. HCl 40.55 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
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