Imidazoline Receptor Imidazoline Receptor

Inhibitor/Activator

Cat.No.	Name	Information
M44871	Harmane	Harmane, a β-Carboline alkaloid (BCA), is a potent neurotoxin that causes severe action tremors and psychiatric manifestations. Harmane is also a potent and selective inhibitor of monoamine oxidase (MAO) (IC50s=0.5 and 5 μM for human MAO A/B, respectively).
M13997	Allantoin	Allantoin is a skin conditioning agent that promotes healthy skin, stimulates new and healthy tissue growth.
M6415	Agmatine sulfate	Agmatine sulfate is an endogenous agonist at imidazoline receptor and a NO synthase inhibitor. Agmatine sulfate exerts modulatory action at multiple molecular targets, such as neurotransmitter systems, ion channels and nitric oxide synthesis.
M5801	Moxonidine	Moxonidine is a selective agonist at the imidazoline receptor subtype 1, used as antihypertensive agent.
M3655	Rilmenidine Phosphate	Rilmenidine Phosphate is a selective I imidazoline receptor agonist which is used for the treatment of hypertension.
M56816	BU224 hydrochloride	BU224 hydrochloride is a selective and high affinity imidazoline I2 receptor ligand, with a Ki of 2.1 nM.
M56815	AGN 192403 hydrochloride	AGN 192403 (BRD4780) hydrochloride is an I1-Imidazoline receptor antagonist for cardiovascular and neurological research.
M42673	RX 801077	RX 801077 (2 BFI free base) is a selective imidazoline I2 receptor (I2R) agonist with a Ki value of 70.1 nM.