Imidazoline Receptor Imidazoline Receptor

Inhibitor/Activator

Cat.No.	Name	Information
M44871	Harmane	Harmane, a β-Carboline alkaloid (BCA), is a potent neurotoxin that causes severe action tremors and psychiatric manifestations. Harmane is also a potent and selective inhibitor of monoamine oxidase (MAO) (IC50s=0.5 and 5 μM for human MAO A/B, respectively).
M13997	Allantoin	Allantoin is a skin conditioning agent that promotes healthy skin, stimulates new and healthy tissue growth.
M6415	Agmatine sulfate	Agmatine sulfate is a α ₂ ligand. Also imidazoline ligand.
M5801	Moxonidine	Moxonidine is a selective agonist at the imidazoline receptor subtype 1, used as antihypertensive agent.
M3655	Rilmenidine Phosphate	Rilmenidine Phosphate is a selective I imidazoline receptor agonist which is used for the treatment of hypertension.
M42673	RX 801077	RX 801077 (2 BFI free base) is a selective imidazoline I2 receptor (I2R) agonist with a Ki value of 70.1 nM.