Inhibitor
| Cat.No. | Name | Information |
|---|---|---|
| M42321 | BMS-502 | BMS-502 is a potent dual inhibitor of diacylglycerol kinase (DGK) α and ζ with IC50 of 4.6 nM and 2.1 nM. |
| M29780 | BAY 2965501 | BAY 2965501 is a potent and selective diacylglycerol kinase zeta (DGKζ) inhibitor that enhances T cell initiation of suboptimal tumor antigens by inhibiting DGKζ. In addition, BAY 2965501 induces pERK activation.BAY 2965501 can be used in cancer research. |
| M50197 | BAY-2862789 | BAY-2862789 is a DGKA inhibitor that can be used in studies related to respiratory diseases and tumors. |
| M49446 | GS-9911 | GS-9911 is a DGKA inhibitor that can be used in studies related to solid tumors. |
| M45317 | (S)-BAY 2965501 | (S)-BAY 2965501 is the left-handed isomer of BAY 2965501 (HY-153343).BAY 2965501 is a potent and selective diacylglycerol kinase zeta (DGKz) inhibitor and induces pERK activation. BAY 2965501 is a potent and selective inhibitor of diacylglycerol kinase zeta (DGKz) and induces pERK activation. |
| M44937 | Momordicine I | Momordicine I, a triterpenoid compound extracted from momordica charantia L. Momordicine I alleviates isoproterenol-induced cardiomyocyte hypertrophy through suppression of PLA2G6 and DGK-ζ. |
| M42327 | DGKζ-IN-1 | DGKζ-IN-1 is an inhibitor of DGKζ. |
| M42326 | AMB639752 | AMB639752 is a potent DGKα inhibitor. |
| M42325 | DGKα-IN-8 | DGKα-IN-8 is a DGKα inhibitor (IC50=22.491 nM; EC50=0.256 nM). |
| M42324 | DGKα-IN-3 | DGKα-IN-3 is a DGKα inhibitor with the IC50 of 283 nM, extracted from patent WO2021105115. |
| M42323 | DGKα-IN-2 | DGKα-IN-2 is a DGKα inhibitor with the IC50 of 0.9 nM, extracted from patent WO2021105115. |
| M42322 | DGKα-IN-4 | DGKα-IN-4 is a DGKα inhibitor with the IC50 of 0.1 nM, extracted from patent WO2021105117. |
| M42320 | DGKα-IN-7 | DGKα-IN-7 is a DGKα inhibitor with the IC50 of 6.225 nM, extracted from patent WO2022271684 (compound 100). |
| M42319 | DGKα-IN-6 | DGKα-IN-6 is a DGKα inhibitor with the IC50 of 1.377 nM, extracted from patent WO2022271650 (compound 143). |
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