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Androgen Receptor Androgen Receptor

Cat.No.  Name Information
M1973 Ostarine (MK-2866) Ostarine (GTx-024 and MK-2866) is an investigational selective androgen receptor modulator (SARM) with Ki of 3.8 nM.
M5565 Dexmedetomidine HCl Dexmedetomidine Hydrochloride is an agonist of adrenergic alpha-2 receptor, which is used in veterinary medicine for its analgesic and sedative properties.
M5805 Nandrolone Nandrolone is a synthetic, anabolic steroid analog of testosterone.
M1839 MDV3100 MDV3100 is an orally bioavailable, organic, non-steroidal small molecule targeting the androgen receptor (AR) with potential antineoplastic activity.
M5764 Medroxyprogesterone acetate Medroxyprogesterone acetate (MPA) is a synthetic progestin and act as a potent progesterone receptor agonist, used to treat abnormal menstruation or irregular vaginal bleeding.
M2270 Apalutamide (ARN-509) Apalutamide (ARN-509) is a novel androgen receptor (AR) antagonist for the treatment of castration-resistant prostate cancer (CRPC).
M10306 Bavdegalutamide (ARV-110) Bavdegalutamide (ARV-110) is an oral, specific androgen receptor (AR) PROTAC degrader.
M3933 Danazol Danazol is a derivative of the synthetic steroid ethisterone that suppresses the production of gonadotrophins and has some weak androgenic effects.
M3750 TAK-700 TAK-700 (Orteronel) is an investigational, oral, nonsteroidal, selective, reversible inhibitor of 17,20-lyase, a key enzyme in the production of androgenic hormones.
M3748 Mestanolone Mestanolone is the 17α-methylated version of dihydrotestosterone (DHT).
M3685 Mesterolone The Mesterolone is an orally applicable androgen, and DHT derivative.
M3428 Stanozolol Stanozolol(Winstrol, Winstrol Depot) is a synthetic anabolic steroid derived from testosterone.
M3234 (R)-Bicalutamide (R)-Bicalutamide is an active competitive non-steroidal androgen receptor antagonist with an IC50 of 0.17 μM for MDA 453 cells.
M3191 Nilutamide Nilutamide (RU 23908) is an androgen receptor (AR) blocker with IC50 of 0.4 μM.
M2910 Oxymetholone Oxymetholone is a 17alpha -alkylated anabolic-androgenic steroid.
M2717 Galeterone Galeterone is a selective CYP17 inhibitor and androgen receptor (AR) antagonist with IC50 of 300 nM and 384 nM, respectively, and is a potent inhibitor of human prostate tumor growth.
M2670 Epiandrosterone Epiandrosterone is a steroid hormone with weak androgenic activity, is a natural metabolite of DHEA.
M2344 RU 58841 RU 58841 is a specific androgen receptor antagonist or anti-androgen.
M2270 Apalutamide (ARN-509) Apalutamide (ARN-509) is a novel androgen receptor (AR) antagonist for the treatment of castration-resistant prostate cancer (CRPC).
M2092 AZD3514 AZD3514 is a potent, orally activie and selective androgen receptor (AR) inhibitor with potential anticancer cancer activity.
M1986 Andarine Andarine (GTx-007, S-4) is a selective nonsteroidal androgen receptor (AR) agonist with Ki of 4 nM.
M1960 Bicalutamide Bicalutamide is an orally active non-steroidal androgen receptor antagonist (IC50 = 190 nM).
M1586 Norelgestromin Norgestimate and its metabolite norelgestromin possess weak androgen-like properties.
M1356 N-Desmethyl Enzalutamide N- Desmethyl Enzalutamide
M57285 Ar-V7-IN-1 Ar-V7-IN-1 is a potent inhibitor of Ar-V7. AR-V7 is a hormone-independent splice variant of the androgen receptor. Ar-V7-IN-1 has the potential for the research of various indications such as prostate cancer.
M57283 SC912 SC912 is a potent and selective AR-V7 inhibitor with IC50 of 0.36 μM. SC912 binds directly to AR-FL and AR-V7 proteins, inhibites nuclear localization and chromatin binding capabilities. SC912 exerts anticancer activity through inhibition of proliferation, induction of cell cycle arrest and apoptosis.
M57282 A4B17 A4B17 is an androgen receptor N-terminal inhibitor, which can be used for the research of androgen-responsive prostate cancer.




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