Cat.No. | Name | Information |
---|---|---|
M1973 | Ostarine (MK-2866) | Ostarine (GTx-024 and MK-2866) is an investigational selective androgen receptor modulator (SARM) with Ki of 3.8 nM. |
M5565 | Dexmedetomidine HCl | Dexmedetomidine Hydrochloride is an agonist of adrenergic alpha-2 receptor, which is used in veterinary medicine for its analgesic and sedative properties. |
M5805 | Nandrolone | Nandrolone is a synthetic, anabolic steroid analog of testosterone. |
M1839 | MDV3100 | MDV3100 is an orally bioavailable, organic, non-steroidal small molecule targeting the androgen receptor (AR) with potential antineoplastic activity. |
M5764 | Medroxyprogesterone acetate | Medroxyprogesterone acetate (MPA) is a synthetic progestin and act as a potent progesterone receptor agonist, used to treat abnormal menstruation or irregular vaginal bleeding. |
M2270 | Apalutamide (ARN-509) | Apalutamide (ARN-509) is a novel androgen receptor (AR) antagonist for the treatment of castration-resistant prostate cancer (CRPC). |
M10306 | Bavdegalutamide (ARV-110) | Bavdegalutamide (ARV-110) is an oral, specific androgen receptor (AR) PROTAC degrader. |
M3933 | Danazol | Danazol is a derivative of the synthetic steroid ethisterone that suppresses the production of gonadotrophins and has some weak androgenic effects. |
M3750 | TAK-700 | TAK-700 (Orteronel) is an investigational, oral, nonsteroidal, selective, reversible inhibitor of 17,20-lyase, a key enzyme in the production of androgenic hormones. |
M3748 | Mestanolone | Mestanolone is the 17α-methylated version of dihydrotestosterone (DHT). |
M3685 | Mesterolone | The Mesterolone is an orally applicable androgen, and DHT derivative. |
M3428 | Stanozolol | Stanozolol(Winstrol, Winstrol Depot) is a synthetic anabolic steroid derived from testosterone. |
M3234 | (R)-Bicalutamide | (R)-Bicalutamide is an active competitive non-steroidal androgen receptor antagonist with an IC50 of 0.17 μM for MDA 453 cells. |
M3191 | Nilutamide | Nilutamide (RU 23908) is an androgen receptor (AR) blocker with IC50 of 0.4 μM. |
M2910 | Oxymetholone | Oxymetholone is a 17alpha -alkylated anabolic-androgenic steroid. |
M2717 | Galeterone | Galeterone is a selective CYP17 inhibitor and androgen receptor (AR) antagonist with IC50 of 300 nM and 384 nM, respectively, and is a potent inhibitor of human prostate tumor growth. |
M2670 | Epiandrosterone | Epiandrosterone is a steroid hormone with weak androgenic activity, is a natural metabolite of DHEA. |
M2344 | RU 58841 | RU 58841 is a specific androgen receptor antagonist or anti-androgen. |
M2270 | Apalutamide (ARN-509) | Apalutamide (ARN-509) is a novel androgen receptor (AR) antagonist for the treatment of castration-resistant prostate cancer (CRPC). |
M2092 | AZD3514 | AZD3514 is a potent, orally activie and selective androgen receptor (AR) inhibitor with potential anticancer cancer activity. |
M1986 | Andarine | Andarine (GTx-007, S-4) is a selective nonsteroidal androgen receptor (AR) agonist with Ki of 4 nM. |
M1960 | Bicalutamide | Bicalutamide is an orally active non-steroidal androgen receptor antagonist (IC50 = 190 nM). |
M1586 | Norelgestromin | Norgestimate and its metabolite norelgestromin possess weak androgen-like properties. |
M1356 | N-Desmethyl Enzalutamide | N- Desmethyl Enzalutamide |
M57285 | Ar-V7-IN-1 | Ar-V7-IN-1 is a potent inhibitor of Ar-V7. AR-V7 is a hormone-independent splice variant of the androgen receptor. Ar-V7-IN-1 has the potential for the research of various indications such as prostate cancer. |
M57283 | SC912 | SC912 is a potent and selective AR-V7 inhibitor with IC50 of 0.36 μM. SC912 binds directly to AR-FL and AR-V7 proteins, inhibites nuclear localization and chromatin binding capabilities. SC912 exerts anticancer activity through inhibition of proliferation, induction of cell cycle arrest and apoptosis. |
M57282 | A4B17 | A4B17 is an androgen receptor N-terminal inhibitor, which can be used for the research of androgen-responsive prostate cancer. |
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