Catalog

Prostaglandin Receptor Prostaglandin Receptor

Inhibitors

Cat.No.	Name	Information
M9473	RO1138452	RO1138452 is a potent and selective antagonist for both human and rat IP receptors and that is possesses analgesic and anti-inflammatory potential.
M9464	Asapiprant	Asapiprant is a potent and selective DP1 receptor antagonist, with a Ki of 0.44 nM.
M9446	Dazoxiben hydrochloride	Dazoxiben hydrochloride is a potent, orally active thromboxane (TX) synthase inhibitor that reduces the formation of blood clots.
M9277	TG4-155	TG4-155 is a brain penetrant prostaglandin EP2 specific antagonist, with a Ki of 9.9 nM.
M9232	PF-04418948	PF-04418948 is a novel, potent and selective prostaglandin EP2 receptor antagonist with IC50 of 16 nM.
M8973	Fevipiprant	Fevipiprant (QAW039) is a selective, potent, reversible competitive CRTh2 antagonist.
M8971	Grapiprant	Grapiprant is a novel, potent and selective prostaglandin EP4 receptor antagonist with antihyperalgesic properties.
M6138	E-7046	E7046 is an orally bioavailable and specific EP4 antagonist, with IC50 of 13.5 nM and Ki of 23.14 nM, exhibiting anti-tumor activities.
M5929	Prostaglandin E2	Prostaglandin E2 is a vasodilator isolated from prostate gland secretion, working by binding and activating the prostaglandin E2 receptor.
M5401	Alprostadil	Alprostadil is used as a drug in the treatment of erectile dysfunction and has vasodilatory properties. It is a Prostaglandin Analog and Prostaglandin E1 Agonist.