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  Catalog
Abmole Inhibitor Catalog 2017

Prostaglandin Receptor Prostaglandin Receptor

Inhibitors

Cat.No.  Name Information
M9776 Darbufelone Darbufelone is a dual inhibitor of cellular PGF2α and LTB4 production, it is also a COX-2 inhibitor potentially for the treatment of rheumatoid arthritis.
M9473 RO1138452 RO1138452 is a potent and selective antagonist for both human and rat IP receptors and that is possesses analgesic and anti-inflammatory potential.
M9464 Asapiprant Asapiprant is a potent and selective DP1 receptor antagonist, with a Ki of 0.44 nM.
M9446 Dazoxiben hydrochloride Dazoxiben hydrochloride is a potent, orally active thromboxane (TX) synthase inhibitor that reduces the formation of blood clots.
M9277 TG4-155 TG4-155 is a brain penetrant prostaglandin EP2 specific antagonist, with a Ki of 9.9 nM.
M9232 PF-04418948 PF-04418948 is a novel, potent and selective prostaglandin EP2 receptor antagonist with IC50 of 16 nM.
M8973 Fevipiprant Fevipiprant (QAW039) is a selective, potent, reversible competitive CRTh2 antagonist.
M8971 Grapiprant Grapiprant is a novel, potent and selective prostaglandin EP4 receptor antagonist with antihyperalgesic properties.
M6138 E-7046 E7046 is an orally bioavailable and specific EP4 antagonist, with IC50 of 13.5 nM and Ki of 23.14 nM, exhibiting anti-tumor activities.
M5929 Prostaglandin E2 Prostaglandin E2 is a vasodilator isolated from prostate gland secretion, working by binding and activating the prostaglandin E2 receptor.
M5401 Alprostadil Alprostadil is used as a drug in the treatment of erectile dysfunction and has vasodilatory properties. It is a Prostaglandin Analog and Prostaglandin E1 Agonist.


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