Inhibitors
Cat.No. | Name | Information |
---|---|---|
M11045 | OR-1896 | Or-1896 is an active longevity metabolite of Levosimendan. Or-1896, a highly selective phosphodiesterase (PDE III) inhibitor, is a powerful vasodilator. |
M10624 | Tetraethylammonium chloride | Tetraethylammonium chloride is a non-selective potassium channel blocker with antitumor properties. |
M10575 | Charybdotoxin TFA | Charybdotoxin TFA, a 37-amino acid peptide, is a K+ channel blocker. |
M10516 | AUT1 | AUT1 is a Kv3 potassium channel modulator which increases whole currents mediated by human Kv3.1b and Kv3.2a channels, with a concomitant leftward shift in the voltage-dependence of activation, while having a less potent effect on hKv3.3 currents. |
M9820 | 2,2,2-Trichloroethanol | 2,2,2-Trichloroethanol is an agonist for the nonclassical K2P channels TREK-1 (KCNK2) and TRAAK (KCNK4). |
M9780 | Nigericin | Nigericin is an antibiotic derived from Streptomyces hygroscopicus, it acts as an H+, K+, Pb2+ ionophore. |
M9700 | ML213 | ML213 (CID-3111211) is a selective KV7.2 (KCNQ2) and KV7.4 (KCNQ4) channel opener, with EC50 values of 230 and 510 nM for KV7.2 and KV7.4, respectively. |
M9423 | CLP290 | CLP290 is a novel, orally available KCC2 modulator, highly selective for KCC2 over related Cl- transporters. |
M9394 | BMS-191011 | BMS-191011 is a potent BKCa channel opener (large-conductance Ca2+-activated potassium channel, KCa1.1). |
M7926 | Minoxidil | Minoxidil activates ATP-activated K+ channels; vasodilator; slow or stop hair loss and promote hair regrowth. |
M7029 | Nigericin sodium salt | Nigericin (NSC 292567) sodium salt is a selective K+ ionophore, Nigericin sodium salt is also an NLRP3 activator which can activate NLRP3 inflammasome to induce pro-inflammatory and immunostimulatory processes. |
M6975 | ML297 | ML297 is a selective Kir3.1/3.2 (GIRK1/2) channel activator. |
M6908 | Linopirdine dihydrochloride | Linopirdine dihydrochloride is a Kv7 (KCNQ) channel blocker. |
M6052 | Vernakalant HCl | Vernakalant Hcl(RSD-1235) is an investigational mixed ion channel blocker that can terminate acute atrial fibrillation (AF) in humans at 2 to 5 mg/kg and may be more atrial-selective than available agents; in treatment of antiarrhythmic. |
M5728 | Lansoprazole | Lansoprazole is a proton-pump inhibitor (PPI) which prevents the stomach from producing gastric acid. |
M5569 | Diazoxide | Diazoxide is a well-known small molecule that activates KATP channels in the smooth muscle of blood vessels and pancreatic beta-cells by increasing membrane permeability to potassium ions. |
M5437 | Azimilide | Azimilide(NE-10064) is a class III antiarrhythmic compound, inhibits I(Ks) and I(Kr) in guinea-pig cardiac myocytes and I(Ks) (minK) channels expressed in Xenopus oocytes. |
M5409 | Amiodarone | Amiodarone HCl is a sodium/potassium-ATPase inhibitor and an autophagy activator, used to treat various types of cardiac dysrhythmias. |
M5368 | 4-Aminopyridine | 4-Aminopyridine is a nonselective K+ channel blocker that binds from the cytoplasmic side of the cell membrane. |
M5302 | ICA069673 | ICA-069673 is a KCNQ2/Q3 potassium channel activator with an IC50 of 0.69 μM. |
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