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Abmole Inhibitor Catalog 2017

Cytochrome P450 (e.g. CYP17) Cytochrome P450 (e.g. CYP17)


Cat.No.  Name Information
M9684 (Rac)-Brassinazole (Rac)-Brassinazole is a brassinosteroid (BR) biosynthesis inhibitor.
M8186 Stiripentol Stiripentol is an LDH inhibitor.
M6451 Apigenin Apigenin is a protein kinase inhibitor.
M6389 1-Aminobenzotriazole (ABT) 1-Aminobenzotriazole (ABT) is a cytochrome P450 inhibitor; inhibits 20-HETE synthesis.
M5650 Fluconazole Fluconazole is a fungal lanosterol 14 alpha-demethylase inhibitor, which thereby prevents the formation of ergosterol,used in the treatment and prevention of superficial and systemic fungal infections.
M5059 Furafylline Furafylline was a potent, non-competitive inhibitor of high affinity phenacetin O-deethylase activity of microsomal fractions of human liver, a reaction catalysed by P450IA2, with an IC50 value of 0.07 microM.
M4146 Sodium-Danshensu Sodium-Danshensu
M4000 Naringenin Naringenin, a common dietary flavonoid abundantly present in fruits and vegetables, is believed to possess strong anti-proliferative properties and the ability to induce apoptosis in hepatoma cell lines.
M3953 Voriconazole Voriconazole is an inhibitor of 14α-lanosterol demethylase with IC50 value of 53nM.
M3708 Anastrozole Anastrozole is a potent and highly selective aromatase (CYP19) inhibitor (IC50 = 15 nM) that has no discernible effect on adrenocorticoid hormone synthesis.
M3591 Abiraterone Acetate Abiraterone Acetate is an acetate salt form of Abiraterone which is a steroidal cytochrome CYP17 inhibitor with IC50 of 72 nM.
M3326 Memantine hydrochloride Memantine hydrochloride is a CYP2B6 and CYP2D6 inhibitor for recombinant CYP2B6 and CYP2D6 with Ki of 0.51 nM and 94.9 μM, respectively.
M2537 Cobicistat Cobicistat (GS-9350) is a potent and selective inhibitor of CYP3A with IC50 of 30-285 nM.
M2058 Ketoconazole Ketoconazole is a potent inhibitor of cytochrome P450c17.
M1839 MDV3100 MDV3100 is an orally bioavailable, organic, non-steroidal small molecule targeting the androgen receptor (AR) with potential antineoplastic activity.
M1814 Avasimibe Avasimibe (CI-1011) is a novel orally bioavailable ACAT inhibitor with IC50 values of 2.9, 13.9, 26.5 µM for CYP2C9, CYP1A2 and CYP2C19, respectively.
M1636 Abiraterone Abiraterone acetate (CB-7598) is a potent, selective, and orally available inhibitor of CYP17 with an IC50 of 4 nM.

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