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  Catalog
Abmole Inhibitor Catalog 2017

Cytochrome P450 (e.g. CYP17) Cytochrome P450 (e.g. CYP17)

Inhibitors

Cat.No.  Name Information
M9931 ε-​Viniferin ε-Viniferin is a potent inhibitor for all the CYP family, with Ki values from 0.5-20 μM.
M9877 Rhapontigenin Rhapontigenin is a selective inactivator of cytochrome P450 1A1 with IC50 of 400 nM.
M9684 (Rac)-Brassinazole (Rac)-Brassinazole is a brassinosteroid (BR) biosynthesis inhibitor.
M8186 Stiripentol Stiripentol is an LDH inhibitor.
M6451 Apigenin Apigenin is a protein kinase inhibitor.
M6389 1-Aminobenzotriazole (ABT) 1-Aminobenzotriazole (ABT) is a cytochrome P450 inhibitor; inhibits 20-HETE synthesis.
M5650 Fluconazole Fluconazole is a fungal lanosterol 14 alpha-demethylase inhibitor, which thereby prevents the formation of ergosterol,used in the treatment and prevention of superficial and systemic fungal infections.
M5059 Furafylline Furafylline was a potent, non-competitive inhibitor of high affinity phenacetin O-deethylase activity of microsomal fractions of human liver, a reaction catalysed by P450IA2, with an IC50 value of 0.07 microM.
M4146 Sodium-Danshensu Danshensu is an active component of Salvia miltiorrhiza (Danshen) that suppresses the formation of reactive oxygen species, inhibits platelet adhesion and aggregation, and protects myocardium against ischemia.
M4000 Naringenin Naringenin, a common dietary flavonoid abundantly present in fruits and vegetables, is believed to possess strong anti-proliferative properties and the ability to induce apoptosis in hepatoma cell lines.
M3953 Voriconazole Voriconazole is an inhibitor of 14α-lanosterol demethylase with IC50 value of 53nM.
M3708 Anastrozole Anastrozole is a potent and highly selective aromatase (CYP19) inhibitor (IC50 = 15 nM) that has no discernible effect on adrenocorticoid hormone synthesis.
M3591 Abiraterone Acetate Abiraterone Acetate is an acetate salt form of Abiraterone which is a steroidal cytochrome CYP17 inhibitor with IC50 of 72 nM.
M3326 Memantine hydrochloride Memantine hydrochloride is a CYP2B6 and CYP2D6 inhibitor for recombinant CYP2B6 and CYP2D6 with Ki of 0.51 nM and 94.9 μM, respectively.
M2537 Cobicistat Cobicistat (GS-9350) is a potent and selective inhibitor of CYP3A with IC50 of 30-285 nM.
M2058 Ketoconazole Ketoconazole is a potent inhibitor of cytochrome P450c17.
M1839 MDV3100 MDV3100 is an orally bioavailable, organic, non-steroidal small molecule targeting the androgen receptor (AR) with potential antineoplastic activity.
M1814 Avasimibe Avasimibe (CI-1011) is a novel orally bioavailable ACAT inhibitor with IC50 values of 2.9, 13.9, 26.5 µM for CYP2C9, CYP1A2 and CYP2C19, respectively.
M1636 Abiraterone Abiraterone acetate (CB-7598) is a potent, selective, and orally available inhibitor of CYP17 with an IC50 of 4 nM.


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