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 About 4 results found for searched term "Tofacitinib" (0.123 seconds)

Cat.No.  Name Target
M1820 Tofacitinib JAK
CP-690550, Tasocitinib
Tofacitinib (formerly tasocitinib, CP-690550) is a novel Janus Kinase 3 (JAK-3) kinase inhibitor with an IC50 value estimated at 0.2 μM.
M3616 Tofacitinib citrate JAK
CP-690550 citrate
Tofacitinib (CP-690550) Citrate is a novel inhibitor of JAK3 with IC50 of 1 nM, 20- to 100-fold less potent against JAK2 and JAK1.
M14324 Tofacitinib metabolite-1 Others
Tofacitinib metabolite-1 is a metabolite of Tofacitinib, a JAK inhibitor. Tofacitinib metabolite-1 can be used in the pharmacokinetics and metabolism studies of tofacitinib.
M27778 (3S,4S)-Tofacitinib JAK
(3S,4S)-Tofacitinib is the less active S-enantiomer of Tofacitinib. Tofacitinib inhibits JAK3 with IC50 of 1 nM.



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