About 5 results found for searched term "CK2-IN-1" (0.08 seconds)
Cat.No. | Name | Target |
---|---|---|
M20381 | WAY-302713-A | Casein Kinase |
CK2α-IN-1 | ||
WAY-302713-A is a selective, non-ATP-competitive CK2α inhibitor (IC50=7.0 µM; Ki=1.6 µM) for cancer-related studies. | ||
M45287 | CK2/ERK8-IN-1 | Casein Kinase |
CK2/ERK8-IN-1 is a dual inhibitor of casein kinase 2 (CK2) (Ki 0.25 µM) and ERK8 (MAPK15, ERK7), both with IC50s of 0.50 µM. In addition, CK2/ERK8-IN-1 binds to PIM1, HIPK2, and DYRK1A with Ki values of 8.65 µM, 15.25 µM, and 11.9 µM, respectively. 15.25 µM and 11.9 µM, respectively, and also has pro-apoptotic activity. | ||
M45293 | BRD4/CK2-IN-1 | Casein Kinase |
BRD4/CK2-IN-1 is a potent, orally active dual-targeted inhibitor of BRD4/CK2 (bromodomain-containing protein 4/casein kinase 2) with IC50 values of 180 nM and 230 nM, respectively.BRD4/CK2-IN-1 exhibits potent anticancer activity without significant toxicity and induces apoptosis and autophagy-related cell death in triple-negative breast cancer (TNBC). autophagy-related cell death in triple negative breast cancer (TNBC). | ||
M45300 | CK2/PIM1-IN-1 | Casein Kinase |
CK2/PIM1-IN-1 is an inhibitor of CK2 and PIM1 with IC50 values of 3.787 μM and 4.327 μM for the effects of CK2 and PIM1, respectively.CAS 번호410483-84-5 | ||
M45312 | CK2-IN-1 | Casein Kinase |
CK2-IN-1 is a CK2 inhibitor with an IC50 value of 150 nM. |
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