About 5 results found for searched term "Aripiprazole" (0.139 seconds)
Cat.No. | Name | Target |
---|---|---|
M3479 | Aripiprazole | 5-HT Receptor |
OPC-14597 | ||
Aripiprazole is a human 5-HT1A receptor partial agonist with a Ki of 4.2 nM. Aripiprazole (OPC-14597) is a potent and high-affinity dopamine D2 receptor partial agonist. | ||
M28078 | Aripiprazole Lauroxil | 5-HT Receptor |
Aripiprazole lauroxil, an N-acyloxymethyl?proagent?of?aripiprazole, is a?Long-acting injectable (LAI)?typical antipsychotic for?schizophrenia. Aripiprazole lauroxil is cleaved by body’s enzyme esterase to N-hydroxymethyl aripiprazole (plus lauric acid) and then to aripiprazole (plus formaldehyde), no toxicity. | ||
M41741 | Dehydroaripiprazole hydrochloride | 5-HT Receptor |
Dehydroaripiprazole (OPC-14857) hydrochloride is an active metabolite of Aripiprazole. | ||
M55458 | Aripiprazole-d8 | 5-HT Receptor |
Aripiprazole-d8 | ||
M28228 | UNC9994 | Dopamine Receptor |
UNC9994, an analog of Aripiprazole, is a functionally selective β-arrestin-biased dopamine D2 receptor (D2R) agonist with EC50 <10 nM for β-arrestin-2 recruitment to D2 receptors. UNC9994 is simultaneously partial agonists of β-arrestin-2 translocation and antagonists of Gi-regulated cAMP production. Antipsychotic Activity. |
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