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Aripiprazole Lauroxil 

Cat. No. M28078

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Aripiprazole Lauroxil  Structure
Size Price Availability Quantity
5mg USD 32  USD32 In stock
10mg USD 50  USD50 In stock
50mg USD 125  USD125 In stock
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Quality Control & Documentation
Biological Activity

Aripiprazole lauroxil, an N-acyloxymethyl?proagent?of?aripiprazole, is a?Long-acting injectable (LAI)?typical antipsychotic for?schizophrenia. Aripiprazole lauroxil is cleaved by body’s enzyme esterase to N-hydroxymethyl aripiprazole (plus lauric acid) and then to aripiprazole (plus formaldehyde), no toxicity.

Chemical Information
Molecular Weight 660.71
Formula C36H51Cl2N3O4
CAS Number 1259305-29-7
Form Solid
Solubility (25°C) DMSO 8.33 mg/mL (ultrasonic)
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Kunal Maini, et al. Neurol Int. Aripiprazole Lauroxil, a Novel Injectable Long-Acting Antipsychotic Treatment for Adults with Schizophrenia: A Comprehensive Review

[2] Roger W Sommi, et al. CNS Spectr. Aripiprazole Lauroxil Dosing Regimens: Understanding Dosage Strengths and Injection Intervals

[3] Adrian Preda, et al. Expert Opin Drug Saf. A safety evaluation of aripiprazole in the treatment of schizophrenia

[4] James E Frampton. Drugs. Aripiprazole Lauroxil: A Review in Schizophrenia

[5] Arpit Aggarwal, et al. Clin Schizophr Relat Psychoses. Aripiprazole Lauroxil Long-Acting Injectable: The Latest Addition to Second-Generation Long-Acting Agents

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Keywords: Aripiprazole Lauroxil  supplier, 5-HT Receptor, inhibitors, activators

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