About 9 results found for searched term "50-44-2" (0.067 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M2744 | GW441756 | Trk |
| GW441756 is a potent, selective inhibitor of TrkA with IC50 of 2 nM, with very little activity to c-Raf1 and CDK2. | ||
| M5771 | Mercaptopurine | DNA/RNA Synthesis |
| 6-MP | ||
| Mercaptopurine (6-MP) inhibits neopurine synthesis by incorporating methyltransferase metabolites of Mercaptopurine into DNA and RNA. | ||
| M7065 | NU9056 | Histone Acetyltransferase |
| NU 9056 | ||
| NU9056 is a potent and selective Tip60 (KAT5) histone acetyltransferase inhibitor with an IC50 of 2 µM. NU9056 shows >16-fold selectivity for Tip60 over PCAF, p300 and GCN5. NU9056 induces apoptosis of prostate cancer cells. | ||
| M8910 | Pamapimod | p38 MAPK |
| R-1503, Ro4402257 | ||
| Pamapimod is a novel p38 mitogen-activated protein kinase inhibitor, inhibited p38alpha and p38beta enzymatic activity, with IC50 values of 0.014 +/- 0.002 and 0.48 +/- 0.04 microM, respectively. | ||
| M11393 | RG7713 | Vasopressin Receptor |
| RO5028442 | ||
| RG7713 (RO5028442) is a highly effective and selective brain-osmotic vasopressin 1A (V1a) receptor antagonist with Ki values of 1 nM (hV1a) and 39 nM (mV1a). | ||
| M13511 | Iberin | Apoptosis |
| NSC 321801 | ||
| Iberin (NSC 321801), a sulfoxide analogue of sulforaphane, is a naturally occurring member of isothiocyanate family. Iberin inhibits cell survival with an IC50 of 2.3 μM in HL60 cell. Iberin induces apoptosis. | ||
| M16643 | Farrerol 7-O-glucoside | Flavonoids |
| Farrerol 7-O-glucoside | ||
| M20385 | WAY-299338 | PDK1 |
| WAY-299338 is a modulator of the Protein Kinase PDK1. | ||
| M42075 | Ruserontinib | EGFR/HER2 |
| Ruserontinib (SKLB1028) is an orally active multikinase inhibitor of EGFR, FLT3 and Abl, with an IC50 value of 55 nM for human FLT3, and has antitumor activity. | ||
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