About 1 result found for searched term "40709-69-1" (0.119 seconds)
Cat.No. | Name | Target |
---|---|---|
M30053 | Bicuculline methiodide | GABA Receptor |
(+)-Bicuculline methiodide; d-Bicuculline methiodide | ||
Bicuculline methiodide is a potent GABA(A) receptors blocker. Bicuculline methiodide alters membrane properties and firing pattern. Bicuculline methiodide reduces the Apamin-sensitive afterhyperpolarization, while Apamin is a toxin isolated from bee venom to block small conductance Ca2+ -activated K+ channels. Bicuculline methiodide facilitates burst firing via blocking apamin-sensitive Ca2+ -activated K+ current. |
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