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XY-06-007 is a selective and potent bump-and-hole (B&H)-PROTAC BRD4BD1L94V degrader. XY-06-007 shows a DC50, 6 h of 10 nM against BRD4BD1L94V with no degradation of off-targets. XY-06-007 demonstrates suitable pharmacokinetics for in vivo studies.
| Molecular Weight | 809.27 |
| Formula | C41H41ClN8O8 |
| CAS Number | 2757045-94-4 |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |
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