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Vanilloid receptor antagonist 1 is a potent vanilloid receptor TRPV1 antagonist.
| Molecular Weight | 305.33 |
| Formula | C18H15N3O2 |
| CAS Number | 871814-52-7 |
| Form | Solid |
| Solubility (25°C) | DMSO 100 mg/mL (ultrasonic) |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[1] Amanda Spring de Almeida, et al. Eur J Pharmacol. TRP channels in cancer pain
[2] Mircea Iftinca, et al. Drugs. TRPV1-Targeted Drugs in Development for Human Pain Conditions
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| 4-ONE
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