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TUG-770

Cat. No. M7541

All AbMole products are for research use only, cannot be used for human consumption.

TUG-770 Structure
Size Price Availability
10mg USD 410  USD410 Out of stock
50mg USD 960  USD960 Out of stock
100mg USD 1500  USD1500 Out of stock
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Quality Control & Documentation
Biological Activity

Tug-770 is a potent, selective, orally active GPR40/FFA1 agonist with an EC50 of 6 nM against human FFA1. Tug-770 has higher selectivity to FFA1 than FFA2, FFA3, FFA4, PPARγ, other receptors, transporters and enzymes.


Chemical Information
Molecular Weight 307.32
Formula C19H14FNO2
CAS Number 1402601-82-4
Solubility (25°C) DMSO ≥ 30 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Christiansen E, et al. ACS Med Chem Lett. Discovery of TUG-770: A Highly Potent Free Fatty Acid Receptor 1 (FFA1/GPR40) Agonist for Treatment of Type 2 Diabetes.

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  Catalog
Abmole Inhibitor Catalog




Keywords: TUG-770 supplier, GPR/FFAR, inhibitors, activators

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