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Terfenadine

Cat. No. M3058

All AbMole products are for research use only, cannot be used for human consumption.

Terfenadine Structure
Synonym:

(±)-Terfenadine; MDL-991

Size Price Availability Quantity
200mg USD 105  USD105 In stock
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Quality Control & Documentation
Biological Activity

Terfenadine is an antihistamine compound that is normally fully metabolized in the liver by the cytochrome P450 CYP3A4 subtype enzyme into the active form fexofenadine.

Chemical Information
Molecular Weight 471.67
Formula C32H41NO2
CAS Number 50679-08-8
Form Solid
Solubility (25°C) DMSO
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Mayra Delgado-Ramrez, et al. Inhibitory effect of terfenadine on Kir2.1 and Kir2.3 channels

[2] D W Aaronson. Effects of terfenadine on psychomotor performance. An overview

[3] J Soto, et al. Terfenadine-induced tremor

[4] R Jankowski, et al. Effect of terfenadine on nasal provocation

[5] H C Masheter. Terfenadine. The first nonsedating antihistamine

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Keywords: Terfenadine, (±)-Terfenadine; MDL-991 supplier, Potassium Channel, inhibitors, activators

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