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TC-G 1004

Cat. No. M7373

All AbMole products are for research use only, cannot be used for human consumption.

TC-G 1004 Structure

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Quality Control & Documentation
Biological Activity

TC-G 1004 is a potent antagonist of adenosine A2A receptors; displays >100-fold selectivity for A2A over A1 receptors (Ki values are 0.44 and 85 nM respectively). Potentiates L-DOPA-induced rotational behavior in 6-OHDA-lesioned rats.

Chemical Information
Molecular Weight 421.5
Formula C22H27N7O2
CAS Number 1061747-72-5
Solubility (25°C) 1eq. HCl 42.15 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Cushing, et al. J Pharmacol Exp Ther. LY215840, a high-affinity 5-HT7 receptor ligand, blocks serotonin-induced relaxation in canine coronary artery.

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Abmole Inhibitor Catalog




Keywords: TC-G 1004 supplier, inhibitors, activators

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