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TC-E 5003

Cat. No. M7365

All AbMole products are for research use only, cannot be used for human consumption.

TC-E 5003 Structure
Synonym:

TCE5003

Size Price Availability Quantity
Free Sample (1-2 mg)  USD 0 In stock
10mM*1mL in DMSO USD 37  USD37 In stock
10mg USD 25  USD25 In stock
25mg USD 39  USD39 In stock
50mg USD 64  USD64 In stock
100mg USD 95  USD95 In stock
200mg USD 135  USD135 In stock
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Quality Control & Documentation
Biological Activity

Tc-e 5003 is a selective inhibitor of PRMT1 with an IC50 of 1.5 µM against hPRMT1. Tc-e 5003 has anti-inflammatory properties in TLR4 signal transduction.

Chemical Information
Molecular Weight 401.26
Formula C16H14Cl2N2O4S
CAS Number 17328-16-4
Solubility (25°C) DMSO 45 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Rowley, et al. J Med Chem. 5-(4-Chlorophenyl)-4-methyl-3-(1-(2-phenylethyl)piperidin-4-yl)isoxazole: a potent, selective antagonist at human cloned dopamine D4 receptors.

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  Catalog
Abmole Inhibitor Catalog




Keywords: TC-E 5003, TCE5003 supplier, PRMTs, inhibitors, activators

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