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Targapremir-210

Cat. No. M27715

All AbMole products are for research use only, cannot be used for human consumption.

Targapremir-210 Structure
Synonym:

TGP-210

Price and Availability

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Quality Control & Documentation
Biological Activity

Targapremir-210 (TGP-210) is a potent and selective miR-210 (miRNA-210, microRNA-210) inhibitor. Targapremir-210 inhibits pre-miR-210 processing with high binding affinity (Kd~200 nM).

Chemical Information
Molecular Weight 592.69
Formula C32H36N10O2
CAS Number 1049722-30-6
Form Solid
Solubility (25°C) DMSO 250 mg/mL (ultrasonic)
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Matthew G Costales, et al. Cell Chem Biol. Targeted Degradation of a Hypoxia-Associated Non-coding RNA Enhances the Selectivity of a Small Molecule Interacting with RNA

[2] Matthew G Costales, et al. J Am Chem Soc. Small Molecule Inhibition of microRNA-210 Reprograms an Oncogenic Hypoxic Circuit

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  Catalog
Abmole Inhibitor Catalog




Keywords: Targapremir-210, TGP-210 supplier, MicroRNA (miRNA), inhibitors, activators

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