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SRPIN803 

Cat. No. M30022

All AbMole products are for research use only, cannot be used for human consumption.

SRPIN803  Structure

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Quality Control & Documentation
Biological Activity

SRPIN803 is a potent CK2 and SRPK1 dual inhibitor, with IC50s of 203 nM and 2.4 μM, respectively. SRPIN803 exhibits antiangiogenic activity. SRPIN803 can be used for the research of age-related macular degeneration.

Chemical Information
Molecular Weight 370.31
Formula C14H9F3N4O3S
CAS Number 380572-02-1
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] George Leonidis, et al. ACS Omega. Synthesis and Biological Evaluation of a c(RGDyK) Peptide Conjugate of SRPIN803

[2] Andrea Dalle Vedove, et al. Eur J Med Chem. A novel class of selective CK2 inhibitors targeting its open hinge conformation

[3] Satoshi Morooka, et al. Mol Pharmacol. Identification of a Dual Inhibitor of SRPK1 and CK2 That Attenuates Pathological Angiogenesis of Macular Degeneration in Mice

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  Catalog
Abmole Inhibitor Catalog




Keywords: SRPIN803  supplier, Casein Kinase, inhibitors, activators

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