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Silmitasertib sodium salt

Cat. No. M13593

All AbMole products are for research use only, cannot be used for human consumption.

Silmitasertib sodium salt Structure
Synonym:

CX-4945 sodium salt

Size Price Availability Quantity
5mg USD 84  USD84 In stock
10mg USD 120  USD120 In stock
25mg USD 240  USD240 In stock
50mg USD 380  USD380 In stock
100mg USD 580  USD580 In stock
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Quality Control & Documentation
Biological Activity

Silmitasertib sodium salt is an orally bioavailable, highly selective and potent CK2 inhibitor, with IC50 values of 1 nM against CK2α and CK2α'.

Chemical Information
Molecular Weight 371.75
CAS Number 1309357-15-0
Solubility (25°C) Water 16.67 mg/mL
DMSO 6.67 mg/mL
Storage 2-8°C, dry, sealed
References

[1] Yuanjiang Wang, et al. J Med Chem. Discovery of 5-(3-Chlorophenylamino)benzo[ c][2,6]naphthyridine Derivatives as Highly Selective CK2 Inhibitors with Potent Cancer Cell Stemness Inhibition

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Keywords: Silmitasertib sodium salt, CX-4945 sodium salt supplier, Casein Kinase, inhibitors, activators

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