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SIAIS164018 hydrochloride

Cat. No. M43432

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SIAIS164018 hydrochloride Structure

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Quality Control & Documentation
Biological Activity

SIAIS164018 hydrochloride is a PROTAC-based ALK and EGFR degrader, with IC50 value of 2.5 nM and 6.6 nM for ALK and ALK G1202R, respectively.

Chemical Information
Molecular Weight 919.79
Formula C43H49Cl2N10O7P
Form Solid
Solubility (25°C) DMSO 75 mg/mL (Need ultrasonic)
Storage 4°C, dry, sealed
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Keywords: SIAIS164018 hydrochloride supplier, PROTAC, inhibitors, activators

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