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Seclidemstat (SP-2577) mesylate is a potent noncompetitive and reversible KDM1A (LSD1) inhibitor (Ki=31 nM, IC50=13 nM). Seclidemstat mesylate promotes antitumor immunity in switch/sucrose nonfermentable (SWI/SNF) complex mutated ovarian cancer, as well as inhibit virus production, viral DNA replication, and late gene expression. Seclidemstat mesylate can be used for the research of Ewing Sarcoma.
| Molecular Weight | 547.04 |
| CAS Number | 2044953-70-8 |
| Solubility (25°C) | DMSO 53.33 mg/mL |
| Storage | 2-8°C, protect from light, dry, sealed |
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