Intepirdine

Cat. No. M3000

All AbMole products are for research use only, cannot be used for human consumption.

Synonym:

GSK 742457; SB-742457; RVT-101

Size	Price	Availability
Free Sample (0.5-1 mg)	USD 0	In stock
1mg	USD 30 USD30	In stock
5mg	USD 60 USD60	In stock
10mg	USD 100 USD100	In stock
25mg	USD 200 USD200	In stock
50mg	USD 300 USD300	In stock

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SB742457 is a highly selective 5-HT6 receptor antagonist with pKi of 9.63, exhibits >100-fold selectivity over other receptors.

	Source	Psychopharmacology (2016). Figure 2. SB742457
	Method	i.v.
	Cell Lines	mice
	Concentrations	3.0 mg/kg
	Incubation Time	30 and 60 min
	Results	In comparison to the vehicle response, there was a significant reduction in glucose solution consumed after the 3.0 mg/kg dose of SB-742457

Molecular Weight	353.44
Formula	C19H19N3O2S
CAS Number	607742-69-8
Solubility (25°C)	DMSO 50 mg/mL
Storage	Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month

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