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RPR132595A hydrochloride

Cat. No. M42331

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RPR132595A hydrochloride Structure

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Quality Control & Documentation
Biological Activity

RPR132595A (NPC) hydrochloride is an active metabolite of CPT-11, which is generated by cytochrome P-450 3A4 (CYP3A4) and finally excreted through urine.

Chemical Information
Molecular Weight 555.02
Formula C28H31ClN4O6
Form Solid
Solubility (25°C) DMSO 50 mg/mL (Need ultrasonic)
Storage 4°C, dry, sealed
References

[1] Semahegn Asemare et al. J Fluoresc. Ground and Excited State Dipole Moments of Metformin Hydrochloride using Solvatochromic Effects and Density Functional Theory

[2] Ha Jung Lee et al. Cells. Nalfurafine Hydrochloride, a κ-Opioid Receptor Agonist, Induces Melanophagy via PKA Inhibition in B16F1 Cells

[3] Chuangchuang Xu et al. Org Biomol Chem. Metal-free and regiospecific synthesis of 3-arylindoles

[4] S Groszkowski et al. Pol J Pharmacol Pharm. 1-Haloacylpiperazines

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Keywords: RPR132595A hydrochloride supplier, Metabolite/Endogenous Metabolite, inhibitors, activators

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