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RLY-2608

Cat. No. M45258

All AbMole products are for research use only, cannot be used for human consumption.

RLY-2608 Structure
Size Price Availability Quantity
1mg USD 630  USD630 In stock
5mg USD 1200  USD1200 In stock
10mg USD 1800  USD1800 In stock
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Quality Control & Documentation
Biological Activity

RLY-2608 is a first-in-class, orally active, selective inhibitor of PI3Ka metabolism.

Chemical Information
Molecular Weight 608.91
Formula C29H14ClF5N6O2
CAS Number 2733573-94-7
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Andreas Varkaris, et al. Cancer Discov. Allosteric PI3Kα Inhibition Overcomes On-target Resistance to Orthosteric Inhibitors Mediated by Secondary PIK3CA Mutations

[2] Andreas Varkaris, et al. Cancer Discov. Discovery and Clinical Proof-of-Concept of RLY-2608, a First-in-Class Mutant-Selective Allosteric PI3Kα Inhibitor That Decouples Antitumor Activity from Hyperinsulinemia

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  Catalog
Abmole Inhibitor Catalog




Keywords: RLY-2608 supplier, PI3K, inhibitors, activators

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