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RGB-286147 

Cat. No. M30608

All AbMole products are for research use only, cannot be used for human consumption.

RGB-286147  Structure

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Quality Control & Documentation
Biological Activity

RGB-286147 is a selective and ATP-competitive CDK and CDK-related kinases (CRK) inhibitor with IC50 values ranging from 9-839 nM. RGB-286147 shows less active against other non-CDK/CRK kinases. RGB-286147 induces cell apoptosis, and exhibits anti-tumor activity.

Chemical Information
Molecular Weight 473.35
Formula C23H22Cl2N4O3
CAS Number 784211-09-2
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Maureen Caligiuri, et al. Chem Biol. A proteome-wide CDK/CRK-specific kinase inhibitor promotes tumor cell death in the absence of cell cycle progression

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  Catalog
Abmole Inhibitor Catalog




Keywords: RGB-286147  supplier, CDK, inhibitors, activators

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