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Relamorelin

Cat. No. M30443

All AbMole products are for research use only, cannot be used for human consumption.

Relamorelin Structure
Synonym:

RM-131; BIM-28131

Price and Availability

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Quality Control & Documentation
Biological Activity

Relamorelin (RM-131), a pentapeptide ghrelin analog, is a selective ghrelin/growth hormone secretagogue receptor (GHSR) agonist with a Ki of 0.42 nM for GHS-1a receptor. Relamorelin is centrally penetrant. Relamorelin increases growth hormone levels and accelerates gastric emptying. Relamorelin has the potential for cachexia, gastroparesis, and gastric/intestinal dysmobility disorders research.

Chemical Information
Molecular Weight 790.97
Formula C43H50N8O5S
CAS Number 661472-41-9
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Rajan Singh, et al. Front Pharmacol. Current Treatment Options and Therapeutic Insights for Gastrointestinal Dysmotility and Functional Gastrointestinal Disorders

[2] Madhusudan Grover, et al. Gut. Gastroparesis: a turning point in understanding and treatment

[3] H Zatorski, et al. J Physiol Pharmacol. Relamorelin and other ghrelin receptor agonists - future options for gastroparesis, functional dyspepsia and proton pump inhibitors-resistant non-erosive reflux disease

[4] Victor Chedid, et al. Expert Opin Investig Drugs. Relamorelin for the treatment of gastrointestinal motility disorders

[5] M Camilleri, et al. Neurogastroenterol Motil. Emerging treatments in Neurogastroenterology: relamorelin: a novel gastrocolokinetic synthetic ghrelin agonist

Related Ghrelin Receptor/GHSR Products
L-692585 

L-692585 is a potent and nonpeptidyl growth hormone secretagogue receptor (GHS-R1a) agonist, with a Ki of 0.8 nM.
PF-6870961 

PF-6870961 is an inverse agonist of GHSR1a with Ki values of 73.6 nM (human GHSR), 239 nM (rat GHSR), and 217 nM (dog GHSR), respectively.
PF-6870961 hydrochloride 

PF-6870961 hydrochloride is an inverse agonist of GHSR1a with Ki values of 73.6 nM (human GHSR), 239 nM (rat GHSR), and 217 nM (dog GHSR), respectively.
des-​Gln14-​Ghrelin

des-Gln14-Ghrelin is a second endogenous ligand for the growth hormone secretagogue receptor.
Obestatin(rat)

Obestatin(rat), encoded by the Ghrelin gene, is a cpeptide, comprised of 23 amino acids.
  Catalog
Abmole Inhibitor Catalog




Keywords: Relamorelin, RM-131; BIM-28131 supplier, Ghrelin Receptor/GHSR, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.


 
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