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Ibutamoren (MK 0677) mesylate is a high affinity ghrelin receptor agonist (pKi = 8.14). Growth hormone (GH) secretagog; stimulates GH release from rat pituitary cells in vitro (EC50 = 1.3 nM) and enhances GH plasma levels in vivo. Also attenuates isoproterenol-induced lipolysis in rat adipocytes in vitro. Orally bioavailable.
| Molecular Weight | 624.77 |
| Formula | C27H36N4O5S.CH3SO3H |
| CAS Number | 159752-10-0 |
| Form | Solid |
| Solubility (25°C) | DMSO 62.48 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
| Related Ghrelin Receptor/GHSR Products |
|---|
| L-692585
L-692585 is a potent and nonpeptidyl growth hormone secretagogue receptor (GHS-R1a) agonist, with a Ki of 0.8 nM. |
| PF-6870961
PF-6870961 is an inverse agonist of GHSR1a with Ki values of 73.6 nM (human GHSR), 239 nM (rat GHSR), and 217 nM (dog GHSR), respectively. |
| PF-6870961 hydrochloride
PF-6870961 hydrochloride is an inverse agonist of GHSR1a with Ki values of 73.6 nM (human GHSR), 239 nM (rat GHSR), and 217 nM (dog GHSR), respectively. |
| des-Gln14-Ghrelin
des-Gln14-Ghrelin is a second endogenous ligand for the growth hormone secretagogue receptor. |
| Obestatin(rat)
Obestatin(rat), encoded by the Ghrelin gene, is a cpeptide, comprised of 23 amino acids. |
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