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Protein kinase inhibitors 1

Cat. No. M9537

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Protein kinase inhibitors 1 Structure
Synonym:

Protein kinase inhibitors I

Size Price Availability Quantity
10mg USD 200  USD200 In stock
25mg USD 450  USD450 In stock
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Biological Activity

Protein kinase inhibitors 1 is a novel inhibitor of HIPK2 with an IC50 of 74 nM and Kd of 9.5 nM.

Chemical Information
Molecular Weight 383.42
Formula C18H17N5O3S
CAS Number 1365986-44-2
Form Solid
Solubility (25°C) DMSO
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Chandrasekhar V Miduturu, et al. Chem Biol. High-throughput Kinase Profiling: A More Efficient Approach Toward the Discovery of New Kinase Inhibitors.

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Keywords: Protein kinase inhibitors 1, Protein kinase inhibitors I supplier, DYRK, inhibitors, activators

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