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Procaine is an inhibitor of sodium channel, NMDA receptor and nAChR with IC50 of 60 μM, 0.296 mM and 45.5 μM, which is also an inhibitor of 5-HT3 with KD of 1.7 μM.
*The compound is unstable in solutions, freshly prepared is recommended
| Molecular Weight | 272.77 |
| Formula | C13H20N2O2.HCl |
| CAS Number | 51-05-8 |
| Solubility (25°C) | DMSO 40 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[1] Thomas Perls. The reappearance of procaine hydrochloride (Gerovital H3) for antiaging
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