Free shipping on all orders over $ 500

Prasugrel

Cat. No. M2234

All AbMole products are for research use only, cannot be used for human consumption.

Prasugrel Structure
Synonym:

Effient, Efient; PCR 4099

Size Price Availability Quantity
50mg USD 30  USD30 In stock
25mg USD 50  USD50 In stock
100mg USD 65  USD65 In stock
200mg USD 95  USD95 In stock
Free Delivery on orders over USD 500 Bulk Inquiry?

Quality Control & Documentation
Biological Activity

Prasugrel is a platelet inhibitor irreversibly binding to P2Y12 receptors. Prasugrel is a member of the thienopyridine class of ADP receptor inhibitors. Prasugrel produces inhibition of platelet aggregation to 20 μM or 5 μM ADP, as measured by light transmission aggregometry.

Chemical Information
Molecular Weight 373.44
Formula C20H20FNO3S
CAS Number 150322-43-3
Solubility (25°C) DMSO 30 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Hyo-Soo Kim, et al. Prasugrel-based de-escalation of dual antiplatelet therapy after percutaneous coronary intervention in patients with acute coronary syndrome (HOST-REDUCE-POLYTECH-ACS): an open-label, multicentre, non-inferiority randomised trial

[2] Marieke Gimbel, et al. Clopidogrel versus ticagrelor or prasugrel in patients aged 70 years or older with non-ST-elevation acute coronary syndrome (POPular AGE): the randomised, open-label, non-inferiority trial

[3] Muhammad Shahzeb Khan, et al. Prasugrel vs. Ticagrelor for Acute Coronary Syndrome Patients Undergoing Percutaneous Coronary Intervention: A Systematic Review and Meta-Analysis

Related P2 Receptor Products
NF449 

NF449 is a highly potent P2X1 receptor antagonist, with IC50s of 0.28, 0.69, and 120 nM for rP2X1, rP2X1+5, P2X2+3, respectively.

NF279 

NF279 is a potent selective and reversible P2X1 receptor antagonist, with an IC50 of 19 nM.

NF110 

NF110 is a P2X3 receptor antagonist (Ki = 36 nM) and inactive toward P2Y receptors stably expressed (IC50s > 10 M).

PSB-12062

PSB-12062 is a potent and selective P2X4 antagonist with an IC50 of 1.38 μM for human P2X4.

NF449 octasodium 

NF449 octasodium is a highly potent P2X1 receptor antagonist, with IC50s of 0.28, 0.69, and 120 nM for rP2X1, rP2X1+5, P2X2+3, respectively.

  Catalog
Abmole Inhibitor Catalog




Keywords: Prasugrel, Effient, Efient; PCR 4099 supplier, P2 Receptor, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.



Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.