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Pim1/AKK1-IN-1

Cat. No. M10227

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Pim1/AKK1-IN-1 Structure
Synonym:

LKB1/AAK1 dual inhibitor

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5mg USD 245  USD245 In stock
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Quality Control & Documentation
Biological Activity

Pim1/AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/75 nM/380 nM for Pim1/AKK1/MST2/LKB1 respectively. Pim1/AKK1-IN-1 also inhibits MPSK1 and TNIK.

Chemical Information
Molecular Weight 339.35
Formula C20H13N5O
CAS Number 1093222-27-5
Solubility (25°C) DMSO 35 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Paul Bamborough, et al. J Med Chem. Assessment of chemical coverage of kinome space and its implications for kinase drug discovery

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  Catalog
Abmole Inhibitor Catalog




Keywords: Pim1/AKK1-IN-1, LKB1/AAK1 dual inhibitor supplier, Pim, inhibitors, activators

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