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Odevixibat (A4250) is a potent selective ileal bile acid transporter (IBAT) inhibitor. Odevixibat (A4250) mitigates cholestatic liver and bile duct damage in mouse models. Odevixibat (A4250) can be used in the study of primary biliary cirrhosis.
| Molecular Weight | 740.93 |
| Formula | C37H48N4O8S2 |
| CAS Number | 501692-44-0 |
| Form | Solid |
| Solubility (25°C) | DMSO ≥ 100 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[2] Emma D Deeks. Drugs. Correction to: Odevixibat: First Approval
[3] Emma D Deeks. Drugs. Odevixibat: First Approval
[4] No authors listed. Am J Health Syst Pharm. Odevixibat Sesquihydrate
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